SCHEMBL7860596

SCHEMBL7860596

O=C(Nc1ccc(N(S)C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1)c1ccccn1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 8/20 0.76
RAF1 P04049 6/20 0.55
KDR P35968 4/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PLK4 O00444 1/20 0.49
CIT O14578 1/20 0.49
AURKA O14965 1/20 0.49
MUSK O15146 1/20 0.49
EPHB6 O15197 1/20 0.49
MAPK13 O15264 1/20 0.49
MLNR O43193 1/20 0.49
MAP3K7 O43318 1/20 0.49
RIPK2 O43353 1/20 0.49
DYRK3 O43781 1/20 0.49
PDE6D O43924 1/20 0.49
NR1I2 O75469 1/20 0.49
STK10 O94804 1/20 0.49
CDK14 O94921 1/20 0.49
ABCB11 O95342 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6815841 0.84 GRM4 (0.51) GRM4RAF1KDRMEN1KMT2A
SCHEMBL7178922 0.83 GRM4 (0.86) GRM4KDRMEN1KMT2AEGFR
SCHEMBL6815923 0.82 IL2 (0.53) GRM4RAF1KDRMEN1KMT2A
SCHEMBL6815329 0.82 KDR (0.56) GRM4RAF1KDRMEN1KMT2A
SCHEMBL6815779 0.78 KDR (0.54) GRM4RAF1KDRMEN1KMT2A
SCHEMBL6810963 0.76 NPC1 (0.50) GRM4MEN1KMT2A
SCHEMBL22216944 0.73 GRM4 (0.76) GRM4KDRMEN1KMT2AHDAC6
SCHEMBL3806472 0.73 KDR (0.53) GRM4KDRMEN1KMT2ACA7
SCHEMBL3275819 0.73 KDR (0.53) GRM4KDRMEN1KMT2ACA7
SCHEMBL11613550 0.73 GRM4 (0.61) GRM4RAF1KDRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137645-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034260-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed