SCHEMBL7861675

SCHEMBL7861675

Cc1cncc(C(=O)Nc2ccccc2)n1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.65
POLB P06746 1/20 0.57
SMN1; SMN2 Q16637 4/20 0.56
CNR1 P21554 5/20 0.55
RAB9A P51151 4/20 0.51
NPC1 O15118 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
CBLB Q13191 1/20 0.49
SCN2A Q99250 1/20 0.49
SCN10A Q9Y5Y9 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
EGFR P00533 1/20 0.49
RECQL P46063 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15006459 0.81 GRM5 (0.47) GRM5POLBSMN1; SMN2CNR1RAB9A
SCHEMBL13201029 0.80 POLB (0.77) GRM5POLBSMN1; SMN2CNR1RAB9A
SCHEMBL30761113 0.80 POLB (0.77) GRM5POLBSMN1; SMN2CNR1RAB9A
SCHEMBL10134797 0.79 CDK2 (0.57) GRM5POLBSMN1; SMN2CNR1RAB9A
SCHEMBL3870458 0.79 GRM5 (1.00) GRM5SMN1; SMN2RAB9ANPC1KDM4E
SCHEMBL10134862 0.76 POLB (0.51) POLBSMN1; SMN2CNR1RAB9ANPC1
SCHEMBL10134912 0.76 POLB (0.51) POLBSMN1; SMN2CNR1RAB9ANPC1
SCHEMBL13097165 0.75 GRM5 (0.54) GRM5POLBCNR1RAB9ANPC1
SCHEMBL22130325 0.75 SMN1; SMN2 (0.72) SMN1; SMN2CNR1RAB9ANPC1KDM4E
SCHEMBL16420803 0.75 IRAK4 (0.63) CNR1RAB9ANPC1SCN2ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128058-A1 DIHYDROPYRIMIDINONES FOR USE AS BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed