SCHEMBL7861738

SCHEMBL7861738

CCOCCn1c(NC2CCNC(Cc3ccc(Cl)c(Cl)c3)C2)nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.43
NR4A2 P43354 1/20 0.43
HRH1 P35367 7/20 0.40
KDM4E B2RXH2 1/20 0.39
IRAK4 Q9NWZ3 2/20 0.38
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861741 1.00 KCNH2 (0.43) KCNH2NR4A2HRH1KDM4EIRAK4
SCHEMBL7854951 0.89 KDM4E (0.45) KCNH2NR4A2HRH1KDM4ECHRM1
SCHEMBL7854950 0.89 KDM4E (0.45) KCNH2NR4A2HRH1KDM4ECHRM1
Oxalic Acid SCHEMBL7864912 0.85 HRH1 (0.45) KCNH2NR4A2HRH1KDM4EIRAK4
Oxalic Acid SCHEMBL7864914 0.85 HRH1 (0.45) KCNH2NR4A2HRH1KDM4EIRAK4
SCHEMBL8713508 0.82 IRAK4 (0.41) HRH1KDM4EIRAK4
SCHEMBL7861794 0.81 TACR1 (0.45) KCNH2HRH1IRAK4
SCHEMBL7861479 0.81 TACR1 (0.45) KCNH2HRH1IRAK4
SCHEMBL7861484 0.81 TACR1 (0.45) KCNH2HRH1IRAK4
SCHEMBL7861787 0.81 TACR1 (0.45) KCNH2HRH1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869955-B1 N-ACYL-2-SUBSTITUTED-4-(BENZIMIDAZOLYL- OR IMIDAZOPYRIDINYL-SUBSTITUTED RESIDUES)-PIPERIDINES AS TACHYKININ ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2001-10-24 EP disclosed