SCHEMBL7862694

SCHEMBL7862694

Cc1cc(C(=O)Nc2ccccc2)n(C)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.59
KMT2A Q03164 6/20 0.55
MEN1 O00255 3/20 0.55
RXFP1 Q9HBX9 1/20 0.54
BRAF P15056 1/20 0.53
ALDH1A1 P00352 3/20 0.51
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
HPGD P15428 1/20 0.51
HIF1A Q16665 1/20 0.51
GAA P10253 2/20 0.51
NAMPT P43490 1/20 0.50
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
KCNJ6 P48051 1/20 0.49
KCNJ5 P48544 1/20 0.49
KCNJ3 P48549 1/20 0.49
AURKA O14965 1/20 0.49
RPS6KB1 P23443 1/20 0.49
CYP1A2 P05177 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664559 0.88 POLB (0.60) TSHRKMT2AMEN1RXFP1ALDH1A1
SCHEMBL17664634 0.87 SMN1; SMN2 (0.59) KMT2AMEN1RXFP1BRAFALDH1A1
SCHEMBL2517076 0.85 KMT2A (0.56) KMT2AMEN1BRAFALDH1A1LMNA
SCHEMBL20852342 0.85 MEN1 (0.55) TSHRKMT2AMEN1RXFP1BRAF
SCHEMBL834743 0.84 KMT2A (0.55) TSHRKMT2AMEN1RXFP1BRAF
SCHEMBL2516724 0.84 KMT2A (0.55) KMT2AMEN1BRAFALDH1A1LMNA
SCHEMBL2517050 0.83 KMT2A (0.48) TSHRKMT2AMEN1RXFP1BRAF
SCHEMBL2874245 0.83 TSHR (0.49) TSHRKMT2AMEN1RXFP1ALDH1A1
SCHEMBL17660199 0.82 GAA (0.54) TSHRKMT2AMEN1RXFP1LMNA
SCHEMBL17660204 0.82 KMT2A (0.53) KMT2AMEN1BRAFALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128058-A1 DIHYDROPYRIMIDINONES FOR USE AS BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed
WO-2008061236-A2 SULFOXIMINES AS KINASE INHIBITORS ALLERGAN, INC. (US) 2008-05-22 WO disclosed