SCHEMBL7862743

SCHEMBL7862743

O=c1c2ccccc2cnn1CCBr

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.62
RAB9A P51151 6/20 0.62
MITF O75030 1/20 0.62
PKM P14618 1/20 0.62
KMT2A Q03164 2/20 0.56
TDP1 Q9NUW8 1/20 0.52
SMN1; SMN2 Q16637 5/20 0.49
LMNA P02545 3/20 0.49
MEN1 O00255 1/20 0.49
GLA P06280 1/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
KDM4E B2RXH2 2/20 0.46
POLB P06746 3/20 0.45
ALDH1A1 P00352 3/20 0.45
MMP2 P08253 1/20 0.44
MMP3 P08254 1/20 0.44
MMP9 P14780 1/20 0.44
MMP13 P45452 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8598953 0.89 NPC1 (0.58) NPC1RAB9AMITFPKMKMT2A
SCHEMBL6216387 0.85 NPC1 (0.64) NPC1RAB9AMITFPKMKMT2A
SCHEMBL10044417 0.83 NPC1 (0.62) NPC1RAB9AMITFPKMKMT2A
SCHEMBL9870217 0.83 NPC1 (0.62) NPC1RAB9AMITFPKMKMT2A
SCHEMBL5108559 0.82 NPC1 (0.65) NPC1RAB9AMITFPKMKMT2A
SCHEMBL29703262 0.81 NPC1 (0.63) NPC1RAB9AMITFPKMKMT2A
SCHEMBL13861649 0.81 NPC1 (0.59) NPC1RAB9AMITFPKMKMT2A
SCHEMBL9382131 0.81 NPC1 (0.63) NPC1RAB9AMITFPKMKMT2A
SCHEMBL3973342 0.80 NPC1 (0.58) NPC1RAB9AMITFPKMKMT2A
SCHEMBL11759940 0.80 NPC1 (0.58) NPC1RAB9AMITFPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923529-B1 SUBSTITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER AG (US) 2001-09-19 EP disclosed
EP-1051403-A1 NOVEL ALKANOIC ACIDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-11-15 EP disclosed
WO-1999038850-A1 NOVEL ALKANOIC ACIDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-08-05 WO disclosed
EP-0923529-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS Bayer Corporation (US) 1999-06-23 EP disclosed
US-5863915-A ENZYME INHIBITORS FOR BONES AND JOINTS BAYER CORPORATION (US) 1999-01-26 US disclosed
WO-1997043237-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER CORPORATION (US) 1997-11-20 WO disclosed