SCHEMBL7866752

SCHEMBL7866752

C=C(c1ccc(S(=O)(=O)NC(C)(C)C)cc1C(F)(F)F)N1CCOc2ccc(-c3ccc4nc(C)[nH]c4c3)cc2C1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 16/20 0.55
PRKDC P78527 1/20 0.39
CREBBP Q92793 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
GPR142 Q7Z601 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3757911 0.92 PIK3CA (0.61) PIK3CAPRKDC
SCHEMBL13054200 0.87 PIK3CA (0.60) PIK3CAPRKDC
SCHEMBL3756702 0.85 PIK3CA (0.62) PIK3CAPRKDCCREBBP
SCHEMBL3750839 0.84 PIK3CA (0.62) PIK3CAPRKDCCREBBPGPR142
SCHEMBL3762172 0.83 PIK3CA (0.60) PIK3CAPRKDC
SCHEMBL3749693 0.83 PIK3CA (0.60) PIK3CAPRKDC
SCHEMBL3753243 0.83 PIK3CA (0.60) PIK3CAPRKDC
SCHEMBL3754069 0.82 PIK3CA (0.72) PIK3CA
SCHEMBL3747696 0.82 PIK3CA (0.59) PIK3CAPRKDC
SCHEMBL13054109 0.79 PIK3CA (0.59) PIK3CAPRKDCCREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed