Iodide

Iodide

SCHEMBL7868477

COc1cc(NC(=O)NC(CN2CCC(CCc3ccc(Cl)c(Cl)c3)CC2)C(C)C)cc(OC)c1OC.I

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 2/20 0.39
CCR3 P51677 6/20 0.74
ALPL P05186 2/20 0.49
ALPI P09923 2/20 0.49
ALPG P10696 2/20 0.49
TP53 P04637 2/20 0.49
POLB P06746 1/20 0.42
BCHE P06276 2/20 0.39
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
KCNH2 Q12809 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1223356 0.92 CCR3 (0.79) CCR3ALPLALPIALPGTP53
SCHEMBL1223352 0.92 CCR3 (0.79) CCR3ALPLALPIALPGTP53
SCHEMBL7865818 0.86 CCR3 (0.76) CCR3ALPLALPIALPGTP53
SCHEMBL5742843 0.84 CCR3 (0.67) CCR3ALPLALPIALPGTP53
SCHEMBL5742848 0.84 CCR3 (0.67) CCR3ALPLALPIALPGTP53
SCHEMBL5854109 0.83 CCR3 (0.66) CCR3ALPLALPIALPGTP53
SCHEMBL5854102 0.83 CCR3 (0.66) CCR3ALPLALPIALPGTP53
SCHEMBL6814195 0.82 CCR3 (0.65) CCR3ALPLALPIALPGTP53
Hydrochloric Acid SCHEMBL5744002 0.81 CCR3 (0.63) CCR3MEN1KMT2AMCHR1
Hydrochloric Acid SCHEMBL5744004 0.81 CCR3 (0.63) CCR3MEN1KMT2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131290-A1 PIPERIDINE CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031033-A1 PIPERIDINE CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed