SCHEMBL7880784

SCHEMBL7880784

CN(C)C(=O)C1CCC(c2cc(N)n3ncc(-c4cn[nH]c4)c3n2)CN1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 15/20 0.46
CCNA2 P20248 13/20 0.46
CDK2 P24941 13/20 0.46
CCNA1 P78396 13/20 0.46
PIK3CA P42336 3/20 0.39
MTOR P42345 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14232237 1.00 CHEK1 (0.46) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL14231717 0.90 CHEK1 (0.48) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL10239412 0.89 CHEK1 (0.50) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL14232420 0.89 CHEK1 (0.47) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL14231723 0.88 CHEK1 (0.46) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL6891872 0.87 CHEK1 (0.62) CHEK1CCNA2CDK2CCNA1
SCHEMBL11931004 0.87 CHEK1 (0.62) CHEK1CCNA2CDK2CCNA1
SCHEMBL14232234 0.85 CHEK1 (0.46) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL14232422 0.85 CHEK1 (0.47) CHEK1CCNA2CDK2CCNA1PIK3CA
SCHEMBL14231721 0.84 CHEK1 (0.49) CHEK1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118207-A1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS SCHERING CORPORATION (US) 2010-10-14 WO disclosed