SCHEMBL7885367

SCHEMBL7885367

N#Cc1cccc(-c2ccc3c(c2)C(=O)C2(CCCC4=C(C=CCC4)C2)C3)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.49
PGR P06401 8/20 0.41
OTUD7B Q6GQQ9 3/20 0.41
HRH3 Q9Y5N1 1/20 0.36
CHEK1 O14757 1/20 0.35
AR P10275 1/20 0.34
CTSD P07339 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7890834 0.86 BACE1 (0.38) BACE1PGROTUD7BAR
SCHEMBL31004 0.86 BACE1 (0.38) BACE1PGROTUD7BAR
SCHEMBL1464867 0.82 BACE1 (0.55) BACE1PGROTUD7BCHEK1
SCHEMBL1464612 0.81 BACE1 (0.60) BACE1PGROTUD7BHRH3CHEK1
SCHEMBL30483 0.80 BACE1 (0.59) BACE1PGROTUD7BHRH3CHEK1
SCHEMBL1465333 0.79 BACE1 (0.52) BACE1PGROTUD7B
SCHEMBL30475 0.78 BACE1 (0.59) BACE1PGROTUD7BCHEK1
SCHEMBL7879908 0.78 TDP1 (0.35)
SCHEMBL12747575 0.77 BACE1 (0.61) BACE1PGROTUD7BHRH3CHEK1
SCHEMBL30303 0.77 BACE1 (0.57) BACE1PGROTUD7BHRH3CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed