SCHEMBL7885484

SCHEMBL7885484

O=c1ccc2cccc(C(c3cccc(C(F)(F)F)c3)n3cncn3)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.40
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
KIF11 P52732 1/20 0.36
AKR1B1 P15121 2/20 0.34
HTT P42858 1/20 0.34
XDH P47989 2/20 0.33
PDE2A O00408 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KCNN4 O15554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7891977 0.83 CYP19A1 (0.44) CYP19A1KIF11HTTCYP3A4CYP2C19
SCHEMBL7885482 0.83 CYP19A1 (0.44) CYP19A1KIF11HTTCYP3A4CYP2C19
Bromide SCHEMBL7885634 0.82 CYP19A1 (0.43) CYP19A1KIF11HTTCYP3A4CYP2C19
Bromide SCHEMBL7885638 0.82 CYP19A1 (0.43) CYP19A1KIF11HTTCYP3A4CYP2C19
SCHEMBL27426144 0.73 CYP19A1 (0.44) CYP19A1CYP3A4CYP2C19
SCHEMBL7893117 0.72 CYP19A1 (0.43) CYP19A1
SCHEMBL7895319 0.72 CYP19A1 (0.43) CYP19A1CYP3A4CYP2C19
Oxalic Acid SCHEMBL27428421 0.71 CNR2 (0.43) CYP19A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10102654 0.71 CYP19A1 (0.40) CYP19A1PDE2AHDAC1HDAC8HDAC6
SCHEMBL7896660 0.71 CYP19A1 (0.46) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800524-B1 6-[TRIAZOLYL[ 3-(TRIFLUOROMETHYL)PHENYL]METHYL]-2-QUINOLINONES AND -QUINOLINETHIONES JANSSEN PHARMACEUTICA NV (BE) 2001-10-31 EP claimed