SCHEMBL7886512

SCHEMBL7886512

COc1cccc(C(C)NC[C@@H]2C[C@H]2c2ccccc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 6/20 0.57
HTR2C P28335 5/20 0.57
HTR2A P28223 3/20 0.50
HTR2B P41595 3/20 0.50
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
FFAR1 O14842 5/20 0.48
KDM1A O60341 3/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
HSD17B2 P37059 1/20 0.47
HTR1A P08908 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
SLC6A2 P23975 1/20 0.46
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
OPRM1 P35372 1/20 0.46
DRD3 P35462 1/20 0.46
OPRK1 P41145 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7884900 1.00 CASR (0.57) CASRHTR2CHTR2AHTR2BDRD2
SCHEMBL7884899 1.00 CASR (0.57) CASRHTR2CHTR2AHTR2BDRD2
SCHEMBL7886595 0.89 HTR2C (0.49) CASRHTR2CHTR2AHTR2BFFAR1
SCHEMBL7886585 0.89 HTR2C (0.49) CASRHTR2CHTR2AHTR2BFFAR1
SCHEMBL7886592 0.89 HTR2C (0.49) CASRHTR2CHTR2AHTR2BFFAR1
SCHEMBL7884872 0.88 HTR2C (0.54) CASRHTR2CHTR2AFFAR1
SCHEMBL8002998 0.88 HTR2C (0.54) CASRHTR2CHTR2AFFAR1
SCHEMBL7884869 0.88 HTR2C (0.54) CASRHTR2CHTR2AFFAR1
SCHEMBL7879525 0.87 HTR2C (0.52) CASRHTR2CHTR2AHTR2BDRD2
SCHEMBL7879524 0.87 HTR2C (0.52) CASRHTR2CHTR2AHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172091-B1 METABOLIC CALCIUM IMBALANCE AND OSTEOPOROSIS ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-01-09 US disclosed
WO-2000021910-A2 1,2-DISUBSTITUTED CYCLOPROPANES ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-04-20 WO disclosed