SCHEMBL789397

SCHEMBL789397

Brc1ccc2nc(NCCCN3CCOCC3)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.51
FLT3 P36888 1/20 0.50
LMNA P02545 2/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
GLA P06280 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
RAD52 P43351 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
HTR1A P08908 4/20 0.48
PIM1 P11309 1/20 0.47
TSHR P16473 3/20 0.47
ACP1 P24666 1/20 0.46
SIGMAR1 Q99720 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5498332 0.93 EGFR (0.49) EGFRLMNAKDM4ENPC1POLB
SCHEMBL8695046 0.83 NPSR1 (0.63) LMNAKDM4ENPC1GLAPOLB
Hydrochloric Acid SCHEMBL8692152 0.81 NPSR1 (0.62) LMNAKDM4ENPC1GLAPOLB
SCHEMBL5491242 0.81 EGFR (0.58) EGFRFLT3LMNAKDM4ENPC1
SCHEMBL1255024 0.79 TSHR (0.57) EGFRLMNAKDM4ENPC1GLA
SCHEMBL16620777 0.77 KDM4E (0.51) FLT3KDM4EKMT2AALDH1A1RXFP1
SCHEMBL3114904 0.76 POLB (0.54) EGFRLMNAKDM4ENPC1GLA
SCHEMBL16621319 0.76 MAPK1 (0.46) LMNAKMT2AALDH1A1TSHRSIGMAR1
SCHEMBL5488941 0.74 EGFR (0.56) EGFRLMNAPOLBKMT2ARXFP1
SCHEMBL16621192 0.73 MAPT (0.54) KDM4EPOLBKMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed