SCHEMBL7898523

SCHEMBL7898523

CCC(C)NC(=O)Nc1ccc(-c2nc3c(c(N4CCOC[C@@H]4C)n2)CCNC3)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.50
KCNH2 Q12809 1/20 0.50
CYP3A4 P08684 4/20 0.47
PIK3CA P42336 3/20 0.47
RPTOR Q8N122 3/20 0.45
MLST8 Q9BVC4 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL414002 0.90 MTOR (0.60) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL440538 0.90 MTOR (0.60) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL414130 0.87 MTOR (0.47) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL442792 0.87 MTOR (0.47) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL7903507 0.86 MTOR (0.54) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL442593 0.83 MTOR (0.59) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL412693 0.83 MTOR (0.59) MTORKCNH2CYP3A4PIK3CARPTOR
Hydrochloric Acid SCHEMBL443714 0.82 MTOR (0.58) MTORKCNH2CYP3A4PIK3CARPTOR
Hydrochloric Acid SCHEMBL443713 0.82 MTOR (0.58) MTORKCNH2CYP3A4PIK3CARPTOR
SCHEMBL442536 0.80 MTOR (0.49) MTORKCNH2CYP3A4PIK3CARPTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed