SCHEMBL7904059

SCHEMBL7904059

Cc1cc(Cn2c(C)c(C(=O)NC(c3cccc(F)c3)C3CCC3)c3cccc(F)c3c2=O)[nH]n1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.44
TACR3 P29371 10/20 0.41
SMYD3 Q9H7B4 2/20 0.34
PDE2A O00408 3/20 0.34
OPRL1 P41146 1/20 0.33
CALCRL Q16602 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1364142 1.00 CYP2C9 (0.44) CYP2C9TACR3SMYD3PDE2AOPRL1
SCHEMBL1364043 0.88 CYP2C9 (0.44) CYP2C9TACR3
SCHEMBL1364413 0.86 CYP2C9 (0.45) CYP2C9TACR3PDE2A
SCHEMBL1366995 0.86 CYP2C9 (0.45) CYP2C9TACR3PPARG
SCHEMBL1364305 0.85 CYP2C9 (0.46) CYP2C9TACR3PDE2A
SCHEMBL1364253 0.85 CYP2C9 (0.45) CYP2C9TACR3PDE2APPARG
SCHEMBL1366497 0.85 CYP2C9 (0.43) CYP2C9TACR3PDE2APPARG
SCHEMBL2149840 0.84 CYP2C9 (0.47) CYP2C9TACR3OPRL1PPARG
SCHEMBL11917800 0.84 CYP2C9 (0.47) CYP2C9TACR3OPRL1PPARG
SCHEMBL11917814 0.84 CYP2C9 (0.47) CYP2C9TACR3PDE2AOPRL1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045948-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-04-29 WO disclosed