SCHEMBL7909860

SCHEMBL7909860

Cc1ccc(-n2ncc(C)n2)c(C(=O)N2C[C@@H]3C[C@@H]3CC2CNc2ccc(C(F)(F)F)cn2)n1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 17/20 0.59
HCRTR2 O43614 13/20 0.59
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385150 1.00 HCRTR1 (0.59) HCRTR1HCRTR2CYP3A4
SCHEMBL3387139 0.92 HCRTR1 (0.67) HCRTR1HCRTR2
SCHEMBL3389550 0.92 HCRTR1 (0.57) HCRTR1HCRTR2CYP3A4
SCHEMBL7903176 0.92 HCRTR1 (0.67) HCRTR1HCRTR2
SCHEMBL7912803 0.92 HCRTR1 (0.57) HCRTR1HCRTR2CYP3A4
SCHEMBL3385248 0.88 HCRTR1 (0.54) HCRTR1HCRTR2CYP3A4
SCHEMBL3385620 0.87 HCRTR1 (0.53) HCRTR1HCRTR2CYP3A4
SCHEMBL3385515 0.87 HCRTR1 (0.51) HCRTR1HCRTR2CYP3A4
SCHEMBL3388412 0.86 HCRTR1 (0.52) HCRTR1HCRTR2CYP3A4
SCHEMBL3386651 0.86 HCRTR1 (0.56) HCRTR1HCRTR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063663-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL] METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF GLAXO GROUP LIMITED (GB) 2010-06-10 WO disclosed