SCHEMBL7912839

SCHEMBL7912839

Cc1ccc(-c2ccccc2)c(C(=O)N2C[C@@H]3C[C@@H]3CC2CNc2ccc(C(F)(F)F)cn2)n1

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.73
HCRTR1 O43613 18/20 0.57
HCRTR2 O43614 11/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3388555 1.00 CYP3A4 (0.73) CYP3A4HCRTR1HCRTR2
SCHEMBL3385613 0.93 CYP3A4 (0.63) CYP3A4HCRTR1HCRTR2
SCHEMBL3386459 0.93 CYP3A4 (0.63) CYP3A4HCRTR1HCRTR2
SCHEMBL262353 0.91 HCRTR1 (0.69) CYP3A4HCRTR1HCRTR2
SCHEMBL3385234 0.91 HCRTR1 (0.69) CYP3A4HCRTR1HCRTR2
SCHEMBL7917283 0.90 HCRTR1 (0.62) CYP3A4HCRTR1HCRTR2
SCHEMBL2471240 0.90 HCRTR1 (0.62) CYP3A4HCRTR1HCRTR2
SCHEMBL3387575 0.90 HCRTR1 (0.68) CYP3A4HCRTR1HCRTR2
SCHEMBL3386463 0.90 CYP3A4 (0.59) CYP3A4HCRTR1HCRTR2
SCHEMBL3389215 0.89 HCRTR1 (0.59) CYP3A4HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063663-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL] METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF GLAXO GROUP LIMITED (GB) 2010-06-10 WO disclosed