SCHEMBL7916360

SCHEMBL7916360

Cc1c(C(=O)NC(c2cccc(F)c2)C2CCC2)c2cccc(F)c2c(=O)n1Cc1ccn(C)n1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.44
TACR3 P29371 10/20 0.41
PPARG P37231 1/20 0.33
WDR5 P61964 3/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
SMYD3 Q9H7B4 1/20 0.33
RIPK1 Q13546 1/20 0.33
APLNR P35414 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12149114 1.00 CYP2C9 (0.44) CYP2C9TACR3PPARGWDR5GRIN1
SCHEMBL1366381 0.90 CYP2C9 (0.45) CYP2C9TACR3PPARGWDR5GRIN1
SCHEMBL1364253 0.88 CYP2C9 (0.45) CYP2C9TACR3PPARGGRIN1GRIN2B
SCHEMBL1364576 0.88 CYP2C9 (0.45) CYP2C9TACR3APLNR
SCHEMBL12149136 0.88 CYP2C9 (0.43) CYP2C9TACR3PPARGWDR5
SCHEMBL12149149 0.87 CYP2C9 (0.45) CYP2C9TACR3PPARG
SCHEMBL7911640 0.87 CYP2C9 (0.44) CYP2C9TACR3PPARGWDR5SMYD3
SCHEMBL7913126 0.86 CYP2C9 (0.43) CYP2C9TACR3WDR5RIPK1
SCHEMBL1364148 0.86 CYP2C9 (0.43) CYP2C9TACR3PPARGWDR5
SCHEMBL11917814 0.86 CYP2C9 (0.47) CYP2C9TACR3PPARGRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045948-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-04-29 WO disclosed