SCHEMBL7916607

SCHEMBL7916607

C[C@H]1CC2CSC(N)=N[C@@]2(c2cc(NC(=O)c3cnc(O)cn3)ccc2F)CO1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.82
KCNH2 Q12809 6/20 0.82
CYP2D6 P10635 2/20 0.76
BACE2 Q9Y5Z0 5/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3303031 0.90 BACE1 (1.00) BACE1KCNH2CYP2D6BACE2
SCHEMBL3303027 0.90 BACE1 (1.00) BACE1KCNH2CYP2D6BACE2
SCHEMBL7918916 0.90 BACE1 (1.00) BACE1KCNH2CYP2D6BACE2
SCHEMBL3299922 0.89 BACE1 (0.78) BACE1KCNH2CYP2D6BACE2
SCHEMBL3299913 0.89 BACE1 (0.78) BACE1KCNH2CYP2D6BACE2
SCHEMBL7922799 0.89 BACE1 (0.65) BACE1KCNH2CYP2D6BACE2
SCHEMBL3300625 0.88 BACE1 (0.84) BACE1KCNH2CYP2D6BACE2
SCHEMBL3300619 0.88 BACE1 (0.84) BACE1KCNH2CYP2D6BACE2
SCHEMBL7927124 0.88 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2
SCHEMBL3302996 0.88 BACE1 (0.83) BACE1KCNH2CYP2D6BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed