SCHEMBL7917302

SCHEMBL7917302

SN1CCN(Cc2nc3nc(-c4ccc5[nH]ncc5c4)nc(N4CCOCC4)c3s2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.50
PIK3CG P48736 4/20 0.45
PIK3CD O00329 4/20 0.45
ROCK2 O75116 4/20 0.42
ROCK1 Q13464 3/20 0.42
PKN2 Q16513 2/20 0.42
PRKCH P24723 1/20 0.42
PRKCQ Q04759 1/20 0.42
GRIA1 P42261 3/20 0.42
CYP2C9 P11712 1/20 0.42
CACNG2 Q9Y698 1/20 0.42
PKN1 Q16512 1/20 0.42
DAPK3 O43293 2/20 0.41
RPS6KA3 P51812 2/20 0.41
AURKA O14965 1/20 0.41
CHEK2 O96017 1/20 0.41
CDK1 P06493 1/20 0.41
PRKACA P17612 1/20 0.41
CDK2 P24941 1/20 0.41
MARK3 P27448 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1310382 0.91 PIK3CA (0.54) PIK3CAPIK3CGPIK3CDROCK2ROCK1
SCHEMBL1309310 0.88 PIK3CA (0.56) PIK3CAPIK3CGPIK3CDDAPK3RPS6KA3
SCHEMBL1309797 0.84 PIK3CA (0.64) PIK3CAPIK3CGPIK3CDROCK2DAPK3
SCHEMBL1309232 0.80 PIK3CA (0.49) PIK3CAPIK3CGPIK3CDCYP2C9PARP1
SCHEMBL1308625 0.79 PIK3CA (0.50) PIK3CAPIK3CGPIK3CDMTORPIK3CB
SCHEMBL1309744 0.77 PIK3CD (0.55) PIK3CAPIK3CGPIK3CDCYP2C9DAPK3
SCHEMBL1309577 0.77 PIK3CA (0.60) PIK3CAPIK3CGPIK3CDROCK2ROCK1
SCHEMBL1311475 0.75 PIK3CA (0.49) PIK3CAPIK3CGPIK3CDROCK2DAPK3
SCHEMBL1311947 0.74 PIK3CA (0.73) PIK3CAPIK3CGPIK3CDDAPK3RPS6KA3
SCHEMBL190060 0.74 PIK3CA (0.73) PIK3CAPIK3CGPIK3CDDAPK3RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010052569-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2010-05-14 WO disclosed