SCHEMBL7922191

SCHEMBL7922191

CC1=CC(C(=O)Cl)(c2noc(C)n2)C=CC1c1ccccc1

nearest known ligand 0.30

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.30
ADORA1 P30542 1/20 0.30
P2RX3 P56373 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913506 0.91 ADORA2A (0.31) ADORA2AADORA1P2RX3
SCHEMBL6193114 0.67 CACNA1D (0.35)
SCHEMBL7922195 0.62 ADORA2A (0.37) ADORA2AADORA1
SCHEMBL3780105 0.60 MAPT (0.33)
SCHEMBL7115170 0.58
SCHEMBL1281643 0.57 NPC1 (0.64)
SCHEMBL6677390 0.56 MEN1 (0.31)
SCHEMBL6071954 0.55 CACNA1D (0.30)
SCHEMBL14752348 0.55 KDM5C (0.54)
SCHEMBL6679649 0.55 CACNA1D (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed