SCHEMBL7924424

SCHEMBL7924424

NC1=NC2(c3cc([N+](=O)[O-])ccc3F)COCCC2CS1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.66
CYP2D6 P10635 1/20 0.53
KCNH2 Q12809 1/20 0.53
BACE2 Q9Y5Z0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12391069 0.88 BACE1 (0.58) BACE1CYP2D6KCNH2BACE2
SCHEMBL9913096 0.85 BACE1 (0.69) BACE1CYP2D6KCNH2BACE2
SCHEMBL2619958 0.85 BACE1 (0.56) BACE1BACE2
SCHEMBL3778192 0.85 BACE1 (0.56) BACE1BACE2
SCHEMBL8036998 0.85 BACE1 (0.56) BACE1BACE2
SCHEMBL3302012 0.83 BACE1 (0.45) BACE1CYP2D6KCNH2BACE2
SCHEMBL3302018 0.83 BACE1 (0.45) BACE1CYP2D6KCNH2BACE2
SCHEMBL3302020 0.83 BACE1 (0.45) BACE1CYP2D6KCNH2BACE2
SCHEMBL9913103 0.82 BACE1 (0.67) BACE1CYP2D6KCNH2BACE2
SCHEMBL7922354 0.82 BACE1 (0.67) BACE1CYP2D6KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed