SCHEMBL7926728

SCHEMBL7926728

COC(=O)c1cc(F)c2[nH]ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.49
SLC6A2 P23975 8/20 0.49
SLC6A4 P31645 8/20 0.49
SLC6A3 Q01959 8/20 0.49
KCNH2 Q12809 1/20 0.48
KDM4E B2RXH2 4/20 0.43
POLB P06746 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
GAA P10253 1/20 0.43
NFKB1 P19838 1/20 0.43
XDH P47989 1/20 0.43
GFER P55789 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
FUT7 Q11130 1/20 0.43
CDK8 P49336 1/20 0.43
PTPN11 Q06124 3/20 0.43
ALDH1A1 P00352 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18031228 0.83 CYP3A4 (0.50) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL18031517 0.83 KDM4E (0.53) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL143239 0.83 CDK8 (0.44) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL255939 0.81 NOTUM (0.44) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL30781376 0.81 NOTUM (0.44) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL7920910 0.81 CDK8 (0.46) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL28362761 0.81 KDM4E (0.49) KDM4EPOLBL3MBTL1LMNATDP1
SCHEMBL121721 0.80 CYP2D6 (0.50) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL30460807 0.79 CYP2D6 (0.48) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL18033213 0.79 POLB (0.39) KDM4EPOLBTDP1CDK8PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228868-B1 ANTICARCINOGENIC AND ANTITUMOR AGENTS ABBOTT LABORATORIES 2001-05-08 US disclosed
WO-2000006556-A1 SUBSTITUTED OXAZOLINES AS ANTIPROLIFERATIVE AGENTS ABBOTT LABORATORIES (US) 2000-02-10 WO disclosed