SCHEMBL7929479

SCHEMBL7929479

NC1=NC2(c3cc(NC(=O)c4cnc(OCF)cn4)ccc3F)COC[C@@H](F)C2CS1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.68
BACE2 Q9Y5Z0 15/20 0.68
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2342984 1.00 BACE1 (0.68) BACE1BACE2CYP2D6CYP2C9KCNH2
SCHEMBL1936075 1.00 BACE1 (0.68) BACE1BACE2CYP2D6CYP2C9KCNH2
SCHEMBL1936001 0.92 BACE1 (0.67) BACE1BACE2CYP2D6KCNH2
SCHEMBL9913175 0.92 BACE1 (0.67) BACE1BACE2CYP2D6KCNH2
SCHEMBL7927201 0.92 BACE1 (0.67) BACE1BACE2CYP2D6KCNH2
SCHEMBL1935180 0.90 BACE1 (0.61) BACE1BACE2CYP2D6KCNH2
SCHEMBL2927148 0.90 BACE1 (0.75) BACE1BACE2CYP2D6KCNH2
SCHEMBL2927156 0.90 BACE1 (0.75) BACE1BACE2CYP2D6KCNH2
SCHEMBL2620112 0.90 BACE1 (0.75) BACE1BACE2CYP2D6KCNH2
SCHEMBL2109350 0.87 BACE1 (0.67) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed