SCHEMBL7933007

SCHEMBL7933007

C=C(OC(C)(C)C)n1ccc2cc(CNC)ccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.34
S1PR1 P21453 1/20 0.33
OXER1 Q8TDS5 1/20 0.33
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
SMO Q99835 1/20 0.32
NR1H2 P55055 4/20 0.32
KDR P35968 6/20 0.32
KCNH2 Q12809 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ITK Q08881 1/20 0.31
PIK3CD O00329 1/20 0.31
ABL1 P00519 1/20 0.31
EGFR P00533 1/20 0.31
HCK P08631 1/20 0.31
SRC P12931 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
MTOR P42345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13456554 0.85 KDR (0.42) CHRNA7S1PR1OXER1NR1H2KDR
SCHEMBL8047542 0.72 BRD4 (0.44) CHRNA7S1PR1NR1H2KDRPIK3CD
SCHEMBL3007425 0.72 NR1H2 (0.45) CHRNA7S1PR1HPGDALOX15NR1H2
SCHEMBL13428863 0.72 PIK3CD (0.45) CHRNA7S1PR1OXER1HPGDALOX15
SCHEMBL3047553 0.71 PDCD1 (0.41) CHRNA7S1PR1NR1H2KDRPIK3CD
SCHEMBL1253366 0.70 CHRNA7 (0.50) CHRNA7
SCHEMBL12043978 0.69 PIK3CD (0.44) S1PR1OXER1NR1H2KDRPIK3CD
SCHEMBL1057433 0.69 PIK3CD (0.44) S1PR1OXER1NR1H2KDRPIK3CD
SCHEMBL29658586 0.69 PIK3CD (0.44) S1PR1OXER1NR1H2KDRPIK3CD
SCHEMBL1058348 0.68 PIK3CD (0.44) S1PR1OXER1NR1H2KDRPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010030967-A1 4-ARYLOXYQUINOLIN-2(1H)-ONES AS MTOR KINASE AND PI3 KINASE INHIBITORS, FOR USE AS ANTI-CANCER AGENTS WYETH LLC (US) 2010-03-18 WO disclosed