SCHEMBL7933176

SCHEMBL7933176

Nc1ccc(-c2nccnc2Oc2ccc(C(=O)c3nc4ccccc4[nH]3)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 20/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1304485 0.91 PDE10A (0.70) PDE10A
SCHEMBL1303247 0.91 PDE10A (0.76) PDE10A
SCHEMBL1304465 0.88 PDE10A (0.64) PDE10A
SCHEMBL1304847 0.87 PDE10A (0.63) PDE10A
SCHEMBL1304334 0.85 PDE10A (0.80) PDE10A
SCHEMBL1304492 0.84 PDE10A (0.78) PDE10A
SCHEMBL1304081 0.84 PDE10A (0.80) PDE10A
SCHEMBL1304094 0.83 PDE10A (0.78) PDE10A
SCHEMBL13372872 0.83 PDE10A (0.67) PDE10A
SCHEMBL1304767 0.83 PDE10A (0.66) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364308-B1 PYRAZINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC (US) 2012-10-24 EP disclosed
WO-2010057121-A1 PYRAZINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC. (US) 2010-05-20 WO disclosed