SCHEMBL793424

SCHEMBL793424

O=C(O)N1CC[C@H](Nc2nccc(Nc3nc4ccc(Br)cc4s3)n2)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.54
HCK P08631 9/20 0.54
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
DYRK1A Q13627 1/20 0.41
HPGDS O60760 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CLK1 P49759 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
LRRK2 Q5S007 1/20 0.39
LCK P06239 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL144366 0.81 ITK (0.52) BTKRAB9ANPC1CYP1A2CYP3A4
SCHEMBL144365 0.81 ITK (0.52) BTKRAB9ANPC1CYP1A2CYP3A4
SCHEMBL30248309 0.74 CYP2C19 (0.55) RAB9ANPC1CYP1A2CYP3A4CYP2C9
SCHEMBL30248193 0.74 CYP2C19 (0.55) RAB9ANPC1CYP1A2CYP3A4CYP2C9
SCHEMBL889065 0.72 USP30 (0.53) RAB9ANPC1CYP1A2CYP3A4CYP2C9
SCHEMBL19205330 0.70 BTK (1.00) BTKHCK
SCHEMBL19205442 0.70 BTK (1.00) BTKHCK
SCHEMBL19205329 0.70 BTK (1.00) BTKHCK
SCHEMBL140852 0.70 LCK (0.66) BTKRAB9ANPC1DYRK1ALRRK2
SCHEMBL140851 0.70 LCK (0.66) BTKRAB9ANPC1DYRK1ALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed