SCHEMBL7934608

SCHEMBL7934608

CC(C)Oc1cccc(CC(=O)NCC(c2ccc(Cl)c(Cl)c2)N2CCN(CCc3ccccc3)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.69
CCR3 P51677 4/20 0.47
HTT P42858 1/20 0.44
TACR2 P21452 1/20 0.43
CNR2 P34972 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7934611 0.90 TACR1 (0.56) TACR1CCR3HTTSIGMAR1THRB
SCHEMBL7925929 0.83 TACR1 (0.88) TACR1CCR3
SCHEMBL7989837 0.81 TACR1 (1.00) TACR1CCR3
SCHEMBL7985915 0.73 TACR1 (0.59) TACR1CCR3
SCHEMBL7925934 0.73 TACR1 (0.72) TACR1CCR3
SCHEMBL7989839 0.71 TACR1 (0.81) TACR1CCR3
Hydrochloric Acid SCHEMBL6229648 0.71 TACR1 (0.52) TACR1CCR3TACR2
Hydrochloric Acid SCHEMBL8432074 0.69 TACR1 (0.52) TACR1TACR2CNR2
Hydrochloric Acid SCHEMBL8067085 0.69 TACR1 (0.48) TACR1TACR2
SCHEMBL7926232 0.67 TACR1 (1.00) TACR1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US claimed
US-6235732-B1 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; SKIN DISORDERS BOEHRINGER INGELHEIM KG (DE) 2001-05-22 US disclosed
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US disclosed
US-5985881-A TREATMENT AND PREVENTION OF RESPIRATORY DISORDERS, INFLAMMATORY EYE DISEASES, INFLAMMATORY SKIN DISEASES, INTESTINAL DISORDERS, OTHER INFLAMMATORY DISEASES BOEHRINGER INGELHEIM KG (DE) 1999-11-16 US disclosed
WO-1996008480-A1 NEUROKININ ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1996-03-21 WO disclosed