SCHEMBL7936459

SCHEMBL7936459

COc1ccccc1N1CCN(C(CNCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
CCR3 P51677 4/20 0.50
NPC1 O15118 1/20 0.50
TACR1 P25103 3/20 0.48
MAPT P10636 3/20 0.48
TP53 P04637 3/20 0.48
THRB P10828 2/20 0.48
LMNA P02545 1/20 0.48
HTR1A P08908 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAPK1 P28482 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HSD17B10 Q99714 1/20 0.47
POLB P06746 1/20 0.47
CCR2 P41597 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7926212 0.91 CCR3 (0.54) GAACCR3TACR1HTR1ACCR2
SCHEMBL7989186 0.86 CCR3 (0.49) CCR3TACR1MAPTTP53THRB
SCHEMBL7936518 0.85 CCR3 (0.60) CCR3TACR1
SCHEMBL7938519 0.85 CCR3 (0.48) CCR3TACR1
SCHEMBL7935457 0.85 TACR1 (0.54) GAACCR3NPC1TACR1LMNA
SCHEMBL7932622 0.85 TACR1 (0.54) GAACCR3NPC1TACR1CCR2
SCHEMBL7926197 0.85 CCR3 (0.67) GAACCR3TACR1TP53THRB
SCHEMBL7926217 0.85 CCR3 (0.48) CCR3TACR1CCR2
SCHEMBL7938479 0.84 CCR3 (0.61) CCR3TACR1THRBMEN1KMT2A
SCHEMBL7934653 0.84 CCR3 (0.60) CCR3TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US claimed
US-6235732-B1 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; SKIN DISORDERS BOEHRINGER INGELHEIM KG (DE) 2001-05-22 US disclosed
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US disclosed
US-5985881-A TREATMENT AND PREVENTION OF RESPIRATORY DISORDERS, INFLAMMATORY EYE DISEASES, INFLAMMATORY SKIN DISEASES, INTESTINAL DISORDERS, OTHER INFLAMMATORY DISEASES BOEHRINGER INGELHEIM KG (DE) 1999-11-16 US disclosed
WO-1996008480-A1 NEUROKININ ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 1996-03-21 WO disclosed