SCHEMBL7937574

SCHEMBL7937574

c1ccc2sc(Nc3ccc(Oc4nccnc4C4CCNCC4)cn3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 19/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7939709 0.88 PDE10A (0.62) PDE10A
SCHEMBL1304435 0.84 PDE10A (0.64) PDE10A
SCHEMBL2366771 0.83 PDE10A (0.48) PDE10A
SCHEMBL1304040 0.79 PDE10A (0.66) PDE10A
SCHEMBL13474590 0.78 PDE10A (0.65) PDE10A
SCHEMBL1303317 0.77 PDE10A (0.77) PDE10A
SCHEMBL2367315 0.77 PDE10A (0.63) PDE10A
SCHEMBL13562707 0.76 PDE10A (0.78) PDE10A
SCHEMBL1303821 0.75 PDE10A (0.64) PDE10A
SCHEMBL9985998 0.74 PDE10A (0.70) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364308-B1 PYRAZINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC (US) 2012-10-24 EP disclosed
WO-2010057121-A1 PYRAZINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC. (US) 2010-05-20 WO disclosed