SCHEMBL7938293

SCHEMBL7938293

Nc1ccnc2c1nc(-c1cccnc1)c(=O)n2C1CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 13/20 0.48
ALDH1A1 P00352 8/20 0.48
TSHR P16473 5/20 0.48
ALOX15 P16050 4/20 0.48
CYP2C19 P33261 4/20 0.48
HPGD P15428 4/20 0.48
AKT1 P31749 4/20 0.47
MTOR P42345 4/20 0.47
CYP3A4 P08684 7/20 0.43
CYP2C9 P11712 7/20 0.43
HSD17B10 Q99714 6/20 0.43
CASP1 P29466 5/20 0.43
CASP7 P55210 5/20 0.43
MAPK1 P28482 4/20 0.43
HIF1A Q16665 4/20 0.43
GLA P06280 3/20 0.43
USP2 O75604 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP11B2 P19099 2/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937482 0.86 CYP1A2 (0.46) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7938231 0.82 CYP1A2 (0.60) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7946218 0.82 CYP1A2 (0.60) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7943737 0.81 CYP1A2 (0.57) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7937497 0.81 AKT1 (0.41) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL3223334 0.80 CYP1A2 (0.55) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7946948 0.79 CYP1A2 (0.40) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7938413 0.79 CYP1A2 (0.44) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7944871 0.77 AKT1 (0.38) CYP1A2ALDH1A1TSHRALOX15CYP2C19
SCHEMBL7944111 0.76 CYP1A2 (0.51) CYP1A2ALDH1A1TSHRALOX15HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed