SCHEMBL793847

SCHEMBL793847

c1cc(-c2ncc3nc[nH]c3n2)c[nH]1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.33
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680853 0.78 NPC1 (0.45) MAPK1KDM4EALDH1A1GLAGAA
SCHEMBL845813 0.77 CDK8 (0.37) PPARAMAPK1
Hydrochloric Acid SCHEMBL4456673 0.77 NPC1 (0.44) MAPK1KDM4EALDH1A1GLAGAA
SCHEMBL31547968 0.77 MAPK1 (0.41) MAPK1
SCHEMBL30850541 0.74 PPARA (0.35) PPARAMAPK1
SCHEMBL18725509 0.73 PDK2 (0.31) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL30677345 0.73 QPCT (0.50) MAPK1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30850625 0.73 KDM4E (0.34) MAPK1KDM4EALDH1A1GLAGAA
SCHEMBL30850674 0.73 PIK3CA (0.39) ALDH1A1
SCHEMBL3027716 0.73 QPCT (0.50) MAPK1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616469-A1 INHIBITORS OF PI3K-DELTA AND METHODS OF THEIR USE AND MANUFACTURE Exelixis, Inc. (US) 2013-07-24 EP disclosed
WO-2012037226-A1 INHIBITORS OF PI3K-DELTA AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-03-22 WO disclosed