SCHEMBL7941794

SCHEMBL7941794

Cc1cc2cc(c1OCF)-c1ncncc1-c1cccc(c1)C21N=C(N)c2ncccc21

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.43
KCNH2 Q12809 15/20 0.43
BACE2 Q9Y5Z0 6/20 0.39
CTSD P07339 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3359362 0.88 BACE1 (0.54) BACE1KCNH2BACE2
SCHEMBL3359201 0.83 BACE1 (0.44) BACE1KCNH2BACE2CTSD
SCHEMBL3360850 0.80 BACE1 (0.38) BACE1KCNH2BACE2CTSD
SCHEMBL3357760 0.78 BACE1 (0.53) BACE1KCNH2BACE2
SCHEMBL3357857 0.77 BACE1 (0.62) BACE1KCNH2BACE2
SCHEMBL3358115 0.77 BACE1 (0.58) BACE1KCNH2BACE2CTSD
SCHEMBL3360047 0.73 BACE1 (0.42) BACE1KCNH2BACE2CTSD
SCHEMBL3358036 0.73 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL3360616 0.72 BACE1 (0.49) BACE1KCNH2BACE2CTSD
SCHEMBL3245127 0.70 BACE1 (0.39) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056194-A1 5H-PYRROLO [ 3, 4-B] PYRIDIN DERIVATIVES AND THEIR USE ASTRAZENECA AB (SE) 2010-05-20 WO disclosed