SCHEMBL7941874

SCHEMBL7941874

CC#CCOc1ccc(C(=O)Nc2ccc(F)c(CNc3cccnc3N)c2)nc1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.60
BACE2 Q9Y5Z0 4/20 0.49
APP P05067 1/20 0.46
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7942878 0.89 BACE1 (0.75) BACE1BACE2APP
SCHEMBL12301454 0.89 BACE1 (0.51) BACE1BACE2AURKAAURKB
SCHEMBL7944850 0.88 BACE1 (0.56) BACE1BACE2AURKAAURKB
SCHEMBL7943122 0.87 BACE1 (0.58) BACE1BACE2AURKAAURKB
SCHEMBL7945065 0.87 BACE1 (0.53) BACE1BACE2AURKAAURKB
SCHEMBL7944561 0.86 BACE1 (0.49) BACE1BACE2AURKAAURKB
SCHEMBL7940351 0.86 BACE1 (0.80) BACE1BACE2APPAURKAAURKB
SCHEMBL7942895 0.86 BACE1 (0.62) BACE1BACE2APP
SCHEMBL7935468 0.85 BACE1 (0.48) BACE1BACE2AURKAAURKB
SCHEMBL7941722 0.85 BACE1 (0.51) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010047372-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY 塩野義製薬株式会社 (JP) 2010-04-29 WO disclosed