SCHEMBL794261

SCHEMBL794261

Cc1cccc(NC(=O)N2CCN(c3nc(N)nc4sc(CCc5cccs5)nc34)CC2)c1.Nc1nc(N2CCN(C(=O)c3ccc(Cl)cc3)CC2)c2nc(CCc3cccs3)sc2n1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 12/20 0.56
KCNH2 Q12809 4/20 0.44
CYP3A4 P08684 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
NLRP3 Q96P20 1/20 0.43
P2RY12 Q9H244 3/20 0.42
LIMK2 P53671 1/20 0.40
FAAH O00519 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655360 0.92 PI4KB (0.65) PI4KBKCNH2CYP3A4P2RY12LIMK2
SCHEMBL655111 0.88 PI4KB (0.45) PI4KBKCNH2SMN1; SMN2
SCHEMBL654888 0.79 PI4KB (0.62) PI4KBKCNH2CYP3A4SMN1; SMN2NLRP3
SCHEMBL655147 0.78 PI4KB (0.48) PI4KB
SCHEMBL652076 0.76 PI4KB (0.63) PI4KBKCNH2CYP3A4SMN1; SMN2NLRP3
SCHEMBL653361 0.76 PI4KB (0.65) PI4KBKCNH2SMN1; SMN2
SCHEMBL651832 0.73 HSP90AA1 (0.47) PI4KB
SCHEMBL653385 0.73 PI4KB (0.74) PI4KBKCNH2CYP3A4LIMK2FAAH
SCHEMBL16163392 0.73 PI4KB (0.64) PI4KBKCNH2CYP3A4SMN1; SMN2NLRP3
SCHEMBL17964555 0.73 PI4KB (1.00) PI4KBKCNH2LIMK2FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP disclosed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO disclosed