SCHEMBL7946055

SCHEMBL7946055

CSC(=N)c1cccc(CNC(=O)OC(C)(C)C)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
GLS O94925 2/20 0.41
NAMPT P43490 2/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NQO2 P16083 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
IDO1 P14902 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
BCHE P06276 1/20 0.37
KCNA5 P22460 1/20 0.36
ADORA2A P29274 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1244570 0.83 NPSR1 (0.46) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL17922691 0.82 ADORA2A (0.48) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL3980110 0.82 GRM2 (0.46) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL112919 0.80 NPSR1 (0.49) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL31098475 0.80 KDM4A (0.43) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL15436036 0.79 CYP1A2 (0.56) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL26616825 0.78 NPSR1 (0.49) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL28520175 0.77 ADORA2A (0.47) KDM4ANPSR1GLSNAMPTPOLB
SCHEMBL16551970 0.77 KDM4A (0.41) KDM4ANPSR1GLSNAMPTL3MBTL1
SCHEMBL29510880 0.77 NPSR1 (0.47) KDM4ANPSR1GLSNAMPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010009334-A1 METHOD FOR PREPARING LARGAZOLE ANALOGS AND USES THEREOF COLORADO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-01-21 WO disclosed