SCHEMBL7947673

SCHEMBL7947673

Cc1c(-c2nc3cc(C(F)(F)F)ccc3s2)c2ccc(Br)cc2n1CC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.57
AKR1A1 P14550 4/20 0.57
PTGDR2 Q9Y5Y4 9/20 0.51
ILK Q13418 1/20 0.43
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7205581 0.88 AKR1B1 (0.55) AKR1B1AKR1A1PTGDR2ILK
SCHEMBL7755700 0.86 PTGDR2 (0.65) AKR1B1AKR1A1PTGDR2ILK
SCHEMBL7755971 0.79 PTGDR2 (0.50) AKR1B1AKR1A1PTGDR2ILK
SCHEMBL7755682 0.75 PTGDR2 (0.56) AKR1B1AKR1A1PTGDR2
SCHEMBL444747 0.73 AKR1B1 (1.00) AKR1B1AKR1A1
SCHEMBL317185 0.70 PTGDR2 (0.66) AKR1B1PTGDR2
SCHEMBL7754412 0.69 PTGDR2 (0.56) AKR1B1AKR1A1PTGDR2
SCHEMBL21032143 0.69 PTGDR2 (0.61) AKR1B1PTGDR2
SCHEMBL21032474 0.69 PTGDR2 (0.61) AKR1B1AKR1A1PTGDR2
SCHEMBL2100600 0.67 AKR1B1 (0.53) AKR1B1AKR1A1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001064205-A2 COMPOSITIONS CONTAINING A SUBSTITUTED INDOLEALKANOIC ACID AND AN ANGIOTENSIN CONVERTING ENZYME INHIBITOR THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2001-09-07 WO disclosed