Fandosentan

Fandosentan

SCHEMBL7947757

CCc1cc(C2=C(C(=O)O)N(c3ccccc3C(F)(F)F)S(=O)(=O)c3ccccc32)cc2c1OCO2.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.98
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
LMNA P02545 2/20 0.36
FABP4 P15090 1/20 0.35
ELANE P08246 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fandosentan SCHEMBL795805 0.99 EDNRA (1.00) EDNRAAKR1C3AKR1C2LMNAFABP4
Fandosentan SCHEMBL29388301 0.99 EDNRA (1.00) EDNRAAKR1C3AKR1C2LMNAFABP4
Fandosentan SCHEMBL7547479 0.98 EDNRA (0.98) EDNRAAKR1C3AKR1C2LMNAFABP4
Fandosentan SCHEMBL6541919 0.98 EDNRA (0.98) EDNRAAKR1C3AKR1C2LMNAFABP4
SCHEMBL7985075 0.91 EDNRA (0.82) EDNRAAKR1C3AKR1C2LMNAELANE
Fandosentan SCHEMBL29566018 0.91 EDNRA (0.85) EDNRAAKR1C3AKR1C2LMNAFABP4
Fandosentan SCHEMBL6541921 0.91 EDNRA (0.85) EDNRAAKR1C3AKR1C2LMNAFABP4
Fandosentan SCHEMBL7947761 0.91 EDNRA (0.85) EDNRAAKR1C3AKR1C2LMNAFABP4
SCHEMBL6542463 0.90 EDNRA (0.83) EDNRAAKR1C3AKR1C2LMNAELANE
SCHEMBL6541350 0.88 EDNRA (0.79) EDNRALMNAFABP4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265399-B1 ALKYLATION; CYCLIZATION WARNER-LAMBERT COMPANY 2001-07-24 US claimed