SCHEMBL7948874

SCHEMBL7948874

Cc1c(C(=O)NC(c2cccc(F)c2)C2CC2)c2cccc(F)c2c(=O)n1CC1CCCNC1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.45
TACR3 P29371 10/20 0.42
P2RX3 P56373 1/20 0.37
GHSR Q92847 1/20 0.36
GNRHR P30968 1/20 0.35
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2148944 1.00 CYP2C9 (0.45) CYP2C9TACR3P2RX3GHSRGNRHR
SCHEMBL11917808 0.94 CYP2C9 (0.43) CYP2C9TACR3P2RX3
SCHEMBL11917803 0.94 CYP2C9 (0.43) CYP2C9TACR3P2RX3
SCHEMBL2149057 0.90 CYP2C9 (0.50) CYP2C9TACR3GNRHR
SCHEMBL7952906 0.89 CYP2C9 (0.46) CYP2C9TACR3
SCHEMBL11917812 0.89 CYP2C9 (0.46) CYP2C9TACR3
SCHEMBL2149840 0.88 CYP2C9 (0.47) CYP2C9TACR3GNRHR
SCHEMBL11917807 0.86 CYP2C9 (0.44) CYP2C9TACR3
SCHEMBL11917804 0.86 CYP2C9 (0.44) CYP2C9TACR3
SCHEMBL2149459 0.85 CYP2C9 (0.47) CYP2C9TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed