SCHEMBL7952274

SCHEMBL7952274

Nc1nccc2ccc(C(=O)N[C@@H](CN3C(=O)c4ccccc4C3=O)c3ccccc3)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 3/20 0.51
MAPK1 P28482 6/20 0.42
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
ROCK1 Q13464 3/20 0.39
ROCK2 O75116 3/20 0.39
RPS6KA5 O75582 2/20 0.39
AKT1 P31749 2/20 0.39
GSK3B P49841 2/20 0.39
NEK4 P51957 2/20 0.39
PRKCD Q05655 2/20 0.39
PRKG2 Q13237 2/20 0.39
PRKG1 Q13976 2/20 0.39
PKN2 Q16513 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
MAPK13 O15264 1/20 0.39
DYRK3 O43781 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982560 0.81 F10 (0.52) F10MAPK1ROCK1ROCK2PPARG
SCHEMBL6982556 0.81 F10 (0.52) F10MAPK1ROCK1ROCK2PPARG
SCHEMBL6981248 0.80 F10 (0.54) F10MAPK1NPC1RAB9AROCK1
SCHEMBL7133910 0.78 F10 (0.50) F10MAPK1ALDH1A1ROCK1ROCK2
SCHEMBL6978044 0.77 F10 (0.49) F10MAPK1ROCK1ROCK2RPS6KA5
SCHEMBL6978051 0.77 F10 (0.49) F10MAPK1ROCK1ROCK2RPS6KA5
SCHEMBL6983225 0.75 F10 (0.49) F10MAPK1ROCK1ROCK2RPS6KA5
SCHEMBL6983223 0.74 F10 (0.49) F10MAPK1ROCK1ROCK2
SCHEMBL6978654 0.73 F10 (0.48) F10MAPK1ROCK1ROCK2AKT1
SCHEMBL6978650 0.73 F10 (0.47) F10MAPK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262069-B1 1-amino-7-isoquinoline derivatives as serine protease inhibitors PROTHERICS MOLECULAR DESIGN LIMITED (GB) 2001-07-17 US disclosed