SCHEMBL7952711

SCHEMBL7952711

O=C(O)C1(c2ccnc(-c3cc(C4(C(=O)O)CCCCC4)ccn3)c2)CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.53
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 1/20 0.43
HDAC4 P56524 3/20 0.42
MAP4K4 O95819 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
SELP P16109 3/20 0.38
SELL P14151 2/20 0.38
LMNA P02545 1/20 0.38
LTB4R Q15722 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1492751 0.82 AKR1C1 (0.51) AKR1C1MEN1KMT2ATSHRHDAC4
SCHEMBL31292176 0.80 AKR1C1 (0.49) AKR1C1MEN1KMT2ATSHRMAP4K4
SCHEMBL29514621 0.79 AKR1C1 (0.66) AKR1C1MEN1KMT2ATSHRHDAC4
SCHEMBL1670449 0.79 AKR1C1 (0.47) AKR1C1MEN1KMT2ATSHRHDAC4
SCHEMBL4827944 0.77 AKR1C1 (0.68) AKR1C1MEN1KMT2ATSHRHDAC4
SCHEMBL1669766 0.75 AKR1C1 (0.42) AKR1C1ALDH1A1
SCHEMBL9280861 0.75 AKR1C3 (0.43) AKR1C1MEN1KMT2ATSHR
SCHEMBL23163719 0.74 MEN1 (0.42) AKR1C1MEN1KMT2ATSHRSELP
SCHEMBL66387 0.72 AKR1C1 (0.96) AKR1C1MEN1KMT2ATSHRHDAC4
SCHEMBL19249602 0.72 AKR1C1 (0.96) AKR1C1MEN1KMT2ATSHRHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed
US-5969150-A FLUORESCENT COMPOUNDS FOR MEDICAL DIAGNOSIS, DRUGS AND LABELS OR FUNGICIDES AND VIRICIDES THE ROCKEFELLER UNIVERSITY (US) 1999-10-19 US disclosed
US-5874587-A FLUORESCENCE THE ROCKEFELLER UNIVERSITY (US) 1999-02-23 US disclosed