SCHEMBL7954468

SCHEMBL7954468

CCc1ccc2cc(C3CCNCC3)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QDPR P09417 1/20 0.47
HTR2C P28335 5/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2A6 P11509 1/20 0.46
TLR9 Q9NR96 3/20 0.44
TLR8 Q9NR97 3/20 0.44
TLR7 Q9NYK1 3/20 0.44
SLC6A4 P31645 5/20 0.43
SLC6A2 P23975 4/20 0.43
SLC6A3 Q01959 4/20 0.43
HTR2A P28223 1/20 0.43
HTR7 P34969 1/20 0.43
HTR2B P41595 1/20 0.43
HTR3A P46098 1/20 0.43
HTR4 Q13639 1/20 0.43
DRD2 P14416 1/20 0.42
SLC18A3 Q16572 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KCNH2 Q12809 1/20 0.41
GABRA1 P14867 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Enefexine SCHEMBL499360 0.83 SLC18A3 (0.55) QDPRHTR2CTLR9TLR8TLR7
SCHEMBL11141177 0.82 CYP1A2 (0.47) CYP1A2CYP2A6SLC6A4SLC6A2SLC6A3
SCHEMBL11141169 0.82 CYP1A2 (0.47) CYP1A2CYP2A6SLC6A4SLC6A2SLC6A3
Enefexine SCHEMBL4886231 0.81 SLC18A3 (0.53) QDPRHTR2CTLR9TLR8TLR7
SCHEMBL11138918 0.81 CYP1A2 (0.46) CYP1A2CYP2A6SLC6A4SLC6A2SLC6A3
SCHEMBL11138912 0.81 CYP1A2 (0.46) CYP1A2CYP2A6SLC6A4SLC6A2SLC6A3
SCHEMBL4518387 0.80 HTR2C (0.62) QDPRHTR2CTLR9TLR8TLR7
Hydrochloric Acid SCHEMBL30946017 0.79 HTR2C (0.63) QDPRHTR2CTLR9TLR8TLR7
SCHEMBL11134820 0.78 CYP2C9 (0.48) CYP1A2CYP2A6SLC6A4DRD2
SCHEMBL11134815 0.78 CYP2C9 (0.48) CYP1A2CYP2A6SLC6A4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed