SCHEMBL7954540

SCHEMBL7954540

c1ccc(COc2ccc3c(c2)OCC(c2ccccc2)C3c2ccccc2OCCCCCCCCCCN2CCOCC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.49
ESR2 Q92731 3/20 0.49
NPSR1 Q6W5P4 2/20 0.44
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
MCHR1 Q99705 1/20 0.42
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6895271 0.90 ESR1 (0.61) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
SCHEMBL6898203 0.90 ESR1 (0.61) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
SCHEMBL6899562 0.89 ESR1 (0.62) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
SCHEMBL7055570 0.84 ESR1 (0.69) ESR1ESR2HTTMCHR1
SCHEMBL8173325 0.80 ESR1 (0.59) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
SCHEMBL7509413 0.80 ESR1 (0.76) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
SCHEMBL7504460 0.80 ESR1 (0.76) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL8501561 0.79 ESR1 (0.58) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7953075 0.79 ESR1 (0.75) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL7500496 0.79 ESR1 (0.75) ESR1ESR2NPSR1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316494-B1 FOR THERAPY AND PROPHYLAXIS OF BONE LOSS, OSTEOPOROSIS, CARDIOVASCULAR DISEASES, COGNITIVE DISORDERS, MENOPAUSAL SYMPTOMS, INCONTINENCE, OBESITY, DYSMENORRHEA, DYSFUNCTIONAL UTERINE BLEEDING, ACNE, HIRSUTISM, POST-PARTUM LACTATION NOVO NORDISK A/S (DK) 2001-11-13 US disclosed