SCHEMBL7957935

SCHEMBL7957935

C=C1CC(c2cccc(Cl)c2)Oc2ccc(Br)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.43
PBRM1 Q86U86 1/20 0.41
CYP19A1 P11511 3/20 0.38
LDHA P00338 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CYP3A4 P08684 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
FFAR1 O14842 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAOB P27338 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1825322 0.86 AR (0.58) ARPBRM1CYP19A1LDHANPC1
SCHEMBL1822330 0.85 AR (0.52) ARPBRM1CYP19A1NPC1RAB9A
SCHEMBL4366347 0.73 AR (0.73) ARCYP19A1LDHANPC1RAB9A
SCHEMBL1823377 0.72 AR (0.57) ARPBRM1CYP19A1NPC1RAB9A
SCHEMBL11246346 0.71 MAOB (0.69) ARCYP19A1NPC1RAB9ACYP3A4
SCHEMBL11246350 0.71 MAOB (0.69) ARCYP19A1NPC1RAB9ACYP3A4
SCHEMBL1823831 0.70 AR (0.58) ARPBRM1CYP19A1NPC1RAB9A
SCHEMBL7958698 0.70 AR (0.52) ARCYP19A1LDHANPC1RAB9A
SCHEMBL1820699 0.70 AR (0.74) ARPBRM1CYP19A1NPC1RAB9A
SCHEMBL14053522 0.70 AR (0.74) ARPBRM1CYP19A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed