SCHEMBL7958868

SCHEMBL7958868

O=C(O)COc1cccc2c1CCCC2N1CCCC1c1nc(-c2ccccc2)c(-c2ccccc2)o1

nearest known ligand 0.86

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 15/20 0.86
PTGDR Q13258 2/20 0.40
TBXAS1 P24557 1/20 0.40
PPARD Q03181 1/20 0.40
FABP4 P15090 1/20 0.39
NR4A2 P43354 2/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7491539 1.00 PTGIR (0.86) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL7487580 1.00 PTGIR (0.86) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL6612770 1.00 PTGIR (0.86) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL7494747 1.00 PTGIR (0.86) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL7491325 0.97 PTGIR (0.82) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL7500155 0.97 PTGIR (0.81) PTGIRPTGDRTBXAS1PPARDFABP4
SCHEMBL7496484 0.97 PTGIR (0.81) PTGIRPTGDRFABP4NR4A2RXRA
SCHEMBL7491137 0.94 PTGIR (0.77) PTGIRPTGDRFABP4
SCHEMBL7489789 0.94 PTGIR (0.76) PTGIRPTGDRPPARDRXRARXRB
SCHEMBL7490049 0.90 PTGIR (0.79) PTGIRPPARDNR4A2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300344-B1 FOR THERAPEUTIC AND/OR PROPHYLACTIC TREATMENT OF ARTERIAL OBSTRUCTION, CEREBROVASCULAR DISEASE, HEPATIC CIRRHOSIS, ARTERIOSCLEROSIS, ISCHEMIC HEART DISEASE, RESTENOSIS AFTER PERCUTANEOUS TRANSLUMINAL CORONARY ANGIOPLASTY, HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-09 US disclosed
US-5972965-A USEFUL FOR INHIBITION OF PLATELET AGGREGATION, VASODILATION, ANTIHYPERTENSIVE ACTIVITY AND PROSTAGLANDIN AGONIST FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-26 US disclosed
EP-0842161-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-05-20 EP disclosed
WO-1997003973-A1 4,5-DIARYL OXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-06 WO disclosed