SCHEMBL7961205

SCHEMBL7961205

CN1O[C@@]2(CC([C@H]3CCCc4ccccc43)Oc3ccc(-c4ccc(F)c(C#N)c4)cc32)N=C1N

nearest known ligand 0.47

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947044 1.00 BACE1 (0.47) BACE1
SCHEMBL12245334 1.00 BACE1 (0.47) BACE1
SCHEMBL12245059 1.00 BACE1 (0.47) BACE1
SCHEMBL7956243 0.90 BACE1 (0.41) BACE1
SCHEMBL7958480 0.90 BACE1 (0.41) BACE1
SCHEMBL7957329 0.89 BACE1 (0.51) BACE1
SCHEMBL7964311 0.89 BACE1 (0.51) BACE1
SCHEMBL7966371 0.89 BACE1 (0.51) BACE1
SCHEMBL7957358 0.89 BACE1 (0.51) BACE1
SCHEMBL7962433 0.89 BACE1 (0.51) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
EP-2324032-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2014-10-01 EP disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed