SCHEMBL7961790

SCHEMBL7961790

CN1C(=O)[C@@]2(C[C@]3(CCCOC3)Oc3ccc(-c4cccc(Br)c4)cc32)N=C1N

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.57
CTSD P07339 17/20 0.57
APP P05067 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7957739 1.00 BACE1 (0.57) BACE1CTSDAPP
SCHEMBL12245167 1.00 BACE1 (0.57) BACE1CTSDAPP
SCHEMBL7955992 1.00 BACE1 (0.57) BACE1CTSDAPP
SCHEMBL7947760 0.91 BACE1 (0.58) BACE1CTSDAPP
SCHEMBL7956734 0.91 BACE1 (0.58) BACE1CTSDAPP
SCHEMBL12246917 0.91 BACE1 (0.58) BACE1CTSDAPP
SCHEMBL7949036 0.90 BACE1 (0.67) BACE1CTSD
SCHEMBL7965156 0.90 BACE1 (0.67) BACE1CTSD
SCHEMBL7950555 0.90 BACE1 (0.67) BACE1CTSD
SCHEMBL7959054 0.90 BACE1 (0.70) BACE1CTSDAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed