SCHEMBL7963915

SCHEMBL7963915

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCN(C)CC2)ccc1C(=O)Nc1cccc2[nH]c(NS(C)(=O)=O)nc12

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 2/20 0.35
AVPR2 P30518 3/20 0.34
AVPR1A P37288 3/20 0.34
AVPR1B P47901 2/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MAP3K7 O43318 2/20 0.32
HTR4 Q13639 3/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7970318 0.99 PTK2 (0.34) PTK2AVPR2AVPR1AAVPR1BMEN1
SCHEMBL7965132 0.93 AVPR2 (0.38) PTK2AVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL7963910 0.93 PTK2 (0.33) PTK2MEN1KMT2AMAP3K7IRAK4
Hydrochloric Acid SCHEMBL7967309 0.93 AVPR2 (0.37) PTK2AVPR2AVPR1AAVPR1BMAP3K7
Hydrochloric Acid SCHEMBL7970313 0.92 PTK2 (0.33) PTK2MEN1KMT2AMAP3K7
SCHEMBL7480849 0.92 AVPR2 (0.35) AVPR2AVPR1AAVPR1BMEN1KMT2A
SCHEMBL7978293 0.91 AVPR2 (0.34) AVPR2AVPR1AAVPR1BMAP3K7IRAK4
Hydrochloric Acid SCHEMBL7481449 0.91 AVPR2 (0.35) AVPR2AVPR1AAVPR1BMAP3K7CYP1A2
Hydrochloric Acid SCHEMBL7963628 0.91 AVPR2 (0.34) AVPR2AVPR1AAVPR1BMAP3K7IRAK4
SCHEMBL7964762 0.91 AVPR2 (0.37) AVPR2AVPR1AAVPR1BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed