SCHEMBL7964374

SCHEMBL7964374

Cc1nc2ccccn2c1-c1ccnc(Nc2cnc(C(=O)O)cn2)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.48
BIRC2 Q13490 1/20 0.48
CDK2 P24941 9/20 0.45
CDK4 P11802 5/20 0.45
CCNE1 P24864 4/20 0.45
MAPK8 P45983 1/20 0.45
MAPK10 P53779 1/20 0.45
PIK3C3 Q8NEB9 2/20 0.41
SYK P43405 1/20 0.41
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
PIK3CA P42336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701624 0.90 XIAP (0.49) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL10252168 0.90 XIAP (0.47) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL10252455 0.86 CDK2 (0.45) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL7975067 0.82 CDK2 (0.66) CDK2CDK4CCNE1SYKALDH1A1
SCHEMBL7978508 0.82 CDK2 (0.51) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL700084 0.81 XIAP (0.45) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL7975631 0.81 CDK2 (0.44) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL7975623 0.79 CDK2 (0.43) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL700972 0.78 HDAC6 (0.47) XIAPBIRC2CDK2CDK4CCNE1
SCHEMBL7978465 0.78 CDK2 (0.47) XIAPBIRC2CDK2CDK4CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010009155-A2 FUSED HETEROCYCLYC INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed