SCHEMBL7965150

SCHEMBL7965150

O=C(Nc1ccc(C(F)(F)F)cc1)c1cccc(Oc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.67
GAA P10253 3/20 0.60
RAB9A P51151 1/20 0.57
KDM4E B2RXH2 2/20 0.56
MAPK1 P28482 2/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
NPSR1 Q6W5P4 1/20 0.56
TLR8 Q9NR97 1/20 0.54
TLR7 Q9NYK1 1/20 0.54
ALDH1A1 P00352 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
P2RY1 P47900 5/20 0.51
NTRK1 P04629 1/20 0.50
KDR P35968 2/20 0.48
BRAF P15056 1/20 0.48
MAPK14 Q16539 1/20 0.48
TNNI3K Q59H18 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29497315 0.93 MAPT (0.65) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL29732862 0.93 MAPT (0.65) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL54805 0.93 MAPT (0.65) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL7612444 0.93 MAPT (0.67) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL7605482 0.92 MAPT (0.67) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL7953536 0.92 MAPT (0.69) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL7953393 0.88 MAPT (0.64) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL3841693 0.87 MAPT (0.75) MAPTGAARAB9AKDM4EMAPK1
SCHEMBL27576744 0.86 MAPT (0.54) MAPTGAARAB9AKDM4EL3MBTL1
SCHEMBL8065139 0.84 MAPT (0.72) MAPTGAARAB9AKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271372-B1 REACTING HETEROAROMATIC HALOGEN COMPOUNDS WITH CARBON MONOXIDE AND AROMATIC AMINES IN THE PRESENCE OF A COMPLEX OF PALLADIUM WITH A TRIPHENYLPHOSPHINE AND A BASE OTHER THAN AN AMINE. LONZA AG (CH) 2001-08-07 US disclosed
US-5900484-A FROM HETEROAROMATIC HALOGEN COMPOUNDS AND AROMATIC AMINES AND CARBON MONOXIDE WITH PALLADIUM PHOSPHINE COMPLEX LONZA AG (CH) 1999-05-04 US disclosed