SCHEMBL7966871

SCHEMBL7966871

O=C(N[C@@H]1Cc2ccc(Cn3cc(CO)c(C(F)(F)F)n3)cc2C1)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 17/20 0.63
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ACHE P22303 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12723923 1.00 GRIA2 (0.63) GRIA2CA1CA2ACHE
SCHEMBL1591094 0.86 GRIA2 (0.73) GRIA2
SCHEMBL1591080 0.84 GRIA2 (0.65) GRIA2
SCHEMBL27812897 0.81 GRIA2 (0.65) GRIA2
SCHEMBL1591016 0.80 GRIA2 (0.61) GRIA2
SCHEMBL1591019 0.80 GRIA2 (0.61) GRIA2
SCHEMBL7902024 0.78 CA1 (0.56) CA1CA2ACHE
SCHEMBL7973199 0.78 CA1 (0.56) CA1CA2ACHE
SCHEMBL1590736 0.78 GRIA2 (1.00) GRIA2
SCHEMBL1590739 0.78 GRIA2 (1.00) GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297110-B1 INDANE DERIVATIVES AS AMPA RECEPTOR MODULATORS MERCK SHARP & DOHME (NL) 2015-05-20 EP disclosed
US-8536214-B2 Indane derivatives as AMPA receptor modulators N.V. ORGANON (NL) 2013-09-17 US disclosed
WO-2009147167-A1 INDANE DERIVATIVES AS AMPA RECEPTOR MODULATORS N.V. ORGANON (NL) 2009-12-10 WO disclosed